HIGHLIGHTS
- who: Alicia Foucourt and colleagues from the CNRS, Bâtiment IRC.O.F. rue Tesnière, Mont-Saint-Aignan, France have published the paper: Design and Synthesis of Thiazolo[5,4-f]quinazolines as DYRK1A Inhibitors, Part II, in the Journal: Molecules 2014, 19, 15411-15439 of 15/09/2014
- what: Structures and DYRK1A/1B IC50 values of the five lead compounds identified in this study (ClogP were calculated with Chemdraw V12.0). The five DYRK1B lead compounds described in this work have been characterized in various in_vitro cellular studies and EHT 5372 has showed . . .
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