Predicting the mutation effects of protein-ligand interactions via end-point binding free energy calculations: strategies and analyses

HIGHLIGHTS

  • who: Yang Yu from the Department of Medicinal Chemistry, China Pharmaceutical University have published the research: Predicting the mutation effects of protein-ligand interactions via end-point binding free energy calculations: strategies and analyses, in the Journal: (JOURNAL)
  • what: The authors have systematically assessed the performance of MM/GBSA and MM/ PBSA approaches on the mutated systems with the consideration of different MD simulation times, dielectric constants and entropy effects. In this study, the binding free_energy difference between the mutated and the wild-type systems was reported (u2206u2206G=u2206GMT-u2206GWT).
  • how: The authors . . .

     

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