Synthesis, in vitro α-glucosidase inhibitory activities, and molecular dynamic simulations of novel 4-hydroxyquinolinone-hydrazones as potential antidiabetic agents

HIGHLIGHTS

  • who: Nahal Shayegan from the Tehran University of Medical Sciences, Shiraz, Iran have published the article: Synthesis, in vitro u03b1-glucosidase inhibitory activities, and molecular dynamic simulations of novel 4-hydroxyquinolinone-hydrazones as potential antidiabetic agents, in the Journal: Scientific Reports Scientific Reports
  • what: In continuation of the work to design u03b1-glucosidase inhibitors, compounds 6a-o were designed and synthesized.
  • how: The results showed that 6m and 6l bind to the active_site on the enzyme and compete with the substrate for binding to the active_site.

SUMMARY

    NMR results . . .

     

    Logo ScioWire Beta black

    If you want to have access to all the content you need to log in!

    Thanks :)

    If you don't have an account, you can create one here.

     

Scroll to Top

Add A Knowledge Base Question !

+ = Verify Human or Spambot ?