Tranilast-tyrosine hybrid molecule exhibits dual activity: suppression of epithelial-mesenchymal transition and induction of cytotoxicity in cancer cells

HIGHLIGHTS

  • who: Tranilast and colleagues from the Kumamoto University: Kumamoto Daigaku have published the paper: Tranilast-Tyrosine Hybrid Molecule Exhibits Dual Activity: Suppression of Epithelial-Mesenchymal Transition and Induction of Cytotoxicity in Cancer Cells, in the Journal: (JOURNAL)
  • what: The authors report the synthesis of a new hybrid molecule, tyrosine-conjugated TNL, and its unexpected dual activity against EMT and cell proliferation. The authors designed a hybrid molecule, TNL-T (Fig 1), by conjugating tyrosine to tranilast via a short linker.
  • how: The authors hypothesized that introducing a tyrosine moiety would increase the intracellular . . .

     

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